Purinergic P2Y1 allosteric antagonist
- Catalog number: NT1119
- Alternate name: NA
- Molar activity: 40-50 Ci/mmol; 1.4-1.8 TBq/mmol
- CAS Number (Parent): 870544-59-5
- Storage conditions: -20°C, in ethanol
- Stability: The rate of decomposition is initially less than 1% for 3 months
- Notes: Shipped on dry ice. To inquire about the current price of this product, please mail us your inquiry below.
References
- “Two disparate ligand-binding sites in the human P2Y1 receptor” D. Zhang, Z.-G. Gao, K. Zhang, E. Kiselev, S. Crane, J. Wang, S. Paoletta, C. Yi, L. Ma, W. Zhang, G.W. Han, H. Liu, V. Cherezov, V. Katritch, H. Jiang, R.C. Stevens, K.A. Jacobson, Q. Zhao and B. Wu (2015) Nature 520(7547): 317-321.
- “Discovery of 2-(phenoxypyridine)-3-phenylureas as small molecule P2Y1 antagonists” H. Chao, H. Turdi, T.F. Herpin, J.Y. Roberge, Y. Liu, D.M. Schnur, M.A. Poss, R. Rehfuss, J. Hua, Q. Wu, L.A. Price, L.M. Abell, W.A. Schumacher, J.S. Bostwick, T.E. Steinbacher, A.B. Stewart, M.L. Ogletree, C.S. Huang, M. Chang, A.M. Cacace, M.J. Arcuri, D. Celani, R.R. Wexler and R.M. Lawrence (2013) Journal of Medicinal Chemistry 56(4): 1704-1714.
